Active Substance: Pilocarpine chloride.
Overview
Welcome to Dwaey, specifically on OFTALMOLOSA CUSI PILOCARPINE 3% page.
This medicine contains an important and useful components, as it consists of
Pilocarpine chlorideis available in the market in concentration
Pilocarpine Hydrochloride
CVD, cholelithiasis, biliary tract dz, COPD, chronic bronchitis, concomitant use of beta adrenergic agonist, renal insufficiency, PUD, Parkinson's, hyperthyroidism, urinary tract obstruction Lactation: unknown if drug is distributed into breast milk; use caution
Dry mouth, Sjogren's syndrome
Angle-closure glaucoma; acute iritis, anterior uveitis; hypersensitivity. Pregnancy.
>10% Sweating (29%),Headache (15%),Flushing (8-13%),Chills (3-15%) 1-10% Nervousness (10%),Nausea (6%),Dizziness (>3%),Asthenia (>3%) Frequency Not Defined Confusion,Hypotension,Hypertension,Bradycardia,Tachycardia,Increased airway resistance,Abdominal cramping,Diarrhea,Urinary frequency,Bladder tightness,Decreased visual acuity
3
Pilocarpine is a tertiary parasympathomimetic that directly stimulates cholinergic receptors in the eyes causing pupillary constriction, spasm of accommodation and a transient rise in IOP followed by a fall.
Concomitant admin of 2 miotics may increase risk of toxic reactions. Aminoglycosides, clindamycin, colistin, cyclopropane and halogenated inhalational anaesthetics, quinine, procainamide, lithium and beta-blockers may reduce the efficacy of pilacarpine. Concurrent use with beta-blockers may lead to bradycardia. May prolong the action of suxamethonium. Potentially Fatal: Miotic and ocular hypotensive effect antagonised by anticholinergics. Conduction disturbances with beta-blockers.
Information not available