Active Substance: Betaxolol (as HCl).
Overview
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This medicine contains an important and useful components, as it consists of
Betaxolol (as HCl)is available in the market in concentration
Betaxolol 0.25% Eye prep
DM, renal or hepatic impairment. May mask signs of hypoglycemia & hyperthyroidism. Gradual withdrawal is recommended. Children. Lactation.
Glaucoma, Ocular hypertension
Hypersensitivity. Sinus bradycardia, cardiogenic shock, overt cardiac failure. Pregnancy .
>10% Ocular effects Short term discomfort (<25%) Frequency Not Defined Ocular Blurred vision,Corneal punctate keratitis,Itching and/or foreign body sensation erythema,Inflammation,Ocular pain and/or discharge,Ocular drynes,Photophobia Systemic Bradycardia, congestive heart failure, heart block,Depression, dizziness, headache, insomnia, lethargy, vertigo,Hair loss, hives, toxic epidermal necrolysis Glossitis,Bronchospasm, dyspnea,Increase in signs and symptoms of myasthenia gravis
3
Betaxolol is a cardioselective Beta-blocker which has greater affinity for ?1-receptors and has little or no effect on ?2-receptors. It lacks intrinsic sympathomimetic but has little membrane-stabilising activity. It also causes the reduction of intraocular pressure by decreasing the production of aqueous humour.
Increased risk of bradycardia w/ digitalis glycosides. May cause mydriasis w/ epinephrine. Potential additive effect w/ oral Ca channel blockers, ?-adrenergic blockers, antiarrhythmics (including amiodarone), parasympathomimetics, guanethidine. Increased risk of myocardial depression and hypotension w/ peripheral muscle relaxants (e.g. tubocurarine).
Information not available