LIDOCAINE AGUETTANT 10mg Injection/Solution for

What is LIDOCAINE AGUETTANT 10mg

LIDOCAINE AGUETTANT 10 mg is a sterile injectable solution containing Lidocaine Hydrochloride, a fast-acting local anesthetic of the amide type. It is primarily used to provide local or regional anesthesia during minor surgical procedures, dental work, or other diagnostic interventions. It can also be employed intravenously in controlled medical settings to treat acute ventricular arrhythmias (abnormal heart rhythms).

• Active Ingredient: Lidocaine Hydrochloride 10 mg per mL
• Concentration: 10 mg/mL (each 10 mL ampoule contains 100 mg)
• Pharmacological Class: Local anesthetic and antiarrhythmic agent
• Administration Routes: Intradermal, subcutaneous, intramuscular, intravenous (by healthcare professional only)

It is often chosen for its rapid onset of action and moderate duration of anesthetic effect. Only trained medical personnel should administer this product due to the potential for serious systemic effects if misused.

How to use LIDOCAINE AGUETTANT 10mg

LIDOCAINE AGUETTANT 10 mg should be administered by qualified healthcare professionals under sterile conditions. The method and dose depend on the clinical indication, the procedure, and patient factors.

• Local Infiltration: Injection directly into the tissue to anesthetize a small area
• Nerve Block: Injection near a nerve or nerve plexus for regional anesthesia
• Epidural or Spinal: For anesthesia during labor or surgery (not all Lidocaine formulations are suitable)
• IV Use: For ventricular arrhythmias under strict monitoring in a hospital setting
• Precautions: Always aspirate before injection to avoid intravascular administration

Dose adjustment is necessary in elderly patients, those with hepatic impairment, or cardiac conditions.

Mode of Action LIDOCAINE AGUETTANT 10mg

Lidocaine works by reversibly blocking sodium channels in neuronal cell membranes, which inhibits the initiation and conduction of nerve impulses. When used intravenously for arrhythmias, it suppresses automaticity in the His-Purkinje system and stabilizes cardiac membranes.

• Local Effect: Numbs targeted area by halting nerve signal transmission
• Cardiac Effect: Reduces ectopic pacemaker activity, stabilizing rhythm
• Onset: 45–90 seconds (IV); 2–5 minutes (local infiltration)
• Duration: 30–60 minutes for local anesthesia

Its dual mechanism allows for versatile applications in both anesthesia and emergency cardiac care.

LIDOCAINE AGUETTANT 10mg Interactions LIDOCAINE AGUETTANT 10mg

Lidocaine can interact with several medications, particularly when administered systemically. Monitoring and dose adjustment may be required.

• Antiarrhythmic drugs (e.g., amiodarone, mexiletine): Increased cardiac depressant effects
• Beta-blockers: May decrease lidocaine clearance
• CYP3A4 inhibitors (e.g., erythromycin, ketoconazole): Elevated plasma levels of lidocaine
• Anticonvulsants: May alter the seizure threshold with lidocaine use
• Other local anesthetics: Potentiation of toxic effects if used together

Notify the healthcare provider about all current medications before administration.

Dosage of LIDOCAINE AGUETTANT 10mg

Dosage should be determined by a healthcare provider based on the patient's weight, the area to be anesthetized, and clinical context.

• Local Infiltration: 3–5 mg/kg body weight, not to exceed 300 mg (30 mL of 10 mg/mL)
• Intravenous (antiarrhythmic use): Initial bolus 1–1.5 mg/kg, followed by infusion (maintenance: 1–4 mg/min)
• Pediatric: Lower weight-based doses are used (maximum 3–4 mg/kg)
• Elderly & hepatic impairment: Use reduced dosage to avoid accumulation

Use the lowest effective dose and avoid repeated or prolonged use unless specifically indicated.

Possible side effects of LIDOCAINE AGUETTANT 10mg

Side effects may vary depending on the route of administration. Systemic absorption can lead to serious reactions if used inappropriately.

• Common (local use): Redness, swelling, mild burning or numbness at injection site
• Systemic (IV use or overdose): Dizziness, tinnitus, blurred vision, confusion
• Severe: Seizures, bradycardia, cardiac arrest, respiratory depression
• Allergic Reaction: Rash, itching, anaphylaxis (rare)

Monitoring is essential during and after administration, especially for IV use.

LIDOCAINE AGUETTANT 10mg Contraindications LIDOCAINE AGUETTANT 10mg

• Known hypersensitivity to lidocaine or other amide-type anesthetics
• Severe sinoatrial, AV, or intraventricular block (in absence of pacemaker)
• Severe hepatic dysfunction
• Porphyria
• Hypovolemia or shock (for certain routes)

Use caution in elderly, debilitated patients or those with cardiac or respiratory conditions.

Storage of LIDOCAINE AGUETTANT 10mg

• Store at controlled room temperature (15–25°C or 59–77°F)
• Protect from light and freezing
• Do not use if solution is cloudy or contains particles
• Keep out of reach of children

Discard any unused solution from opened ampoules. Follow local guidelines for safe disposal.